Synthesis and characterization of thiolated β-cyclodextrin as a novel mucoadhesive excipient for intra-oral drug delivery - Abstract

Highlights

•Synthesis and characterization of cysteamine conjugated β-cyclodextrin (β-CD-Cys).

•Conjugates showed no toxic effects on Caco-2 cells at concentrations of 0.5% (m/v).

•Maximum 34.51-fold improved mucoadhesion on the porcine buccal mucosa.

•Inclusion complexes resulted in 150-fold increased water solubility of miconazole nitrate.

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